Products

Our ligands’ value:

  • Potent (Ki < 100 nM) and subtype selective ( > 500-fold).
  • Their fluorophores are stable, guarantee their affinity and display a variety of photo-physical properties that meet the market demand for several applications from competitive binding assays to microscopy
  • Their pharmacophores are representative of the target and aligned with international standards
  • Their spacers allow optimal target recognition and placing of the fluorophore in the outer region of the membrane.

Showing all 15 results

  • CELT- 174

    Potent and selective hD2 Dopamine receptor fluorescent antagonist (589/616)

    Our hD2 Dopamine receptor fluorescent antagonist shows high affinity for hD2 receptor and selectivity over the other receptor subtypes (Ki =1.06 nM for hD2 receptor in radioligand binding assay). It allows to perform cell visualization in fluorescence microscopy, confocal microscopy and high content system experiments. It is potentially suitable for other fluorescence-based assays.

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  • CELT-240

    Potent hD2/D3 Dopamine receptors fluorescent ligand (589/616)

    Our hD3/D2 Dopamine receptors fluorescent ligand shows high affinity for hD2 and hD3 receptors (Ki =2.34 nM and 2.14 nM respectively in radioligand binding assays) and selectivity over D4 dopamine receptor. It allows to perform cell visualization in fluorescence microscopy, confocal microscopy and high content system experiments. It is potentially suitable for other fluorescence-based assays.

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  • CELT-241

    Potent hD2/D3 Dopamine receptors fluorescent ligand (646/662)

    Our hD2/D3 Dopamine receptors fluorescent ligand shows a high affinity for hD2 and hD3 receptors (Ki = 5.22 nM and 4.77 nM respectively in radioligand binding assays) nd selectivity over D4 dopamine receptor. It allows to perform cell visualization in fluorescence microscopy, confocal microscopy and high content system experiments. It is potentially suitable for other fluorescence-based assays.

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  • CELT-298

    Potent Pan Adenosine receptors fluorescent antagonist (646/662)

    Our Pan Adenosine receptors fluorescent antagonist shows affinity for hA1, hA2A, hA2B and hA3 Adenosine receptors (Ki =20.9 nM, 171 nM, 44,7nM and 95.2 nM respectively in radioligand binding assays). It allows to perform cell visualization in fluorescence microscopy, confocal microscopy and high content system experiments. It is potentially suitable for other fluorescence-based assays.

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  • CELT-372

    Potent and partially selective hA1 Adenosine receptors fluorescent antagonist (589/616)

    Our potent and partially selective hA1 Adenosin receptor fluorescent antagonist shows affinity for hA1, hA2A and hA2B Adenosine receptors (Ki =1.89 nM, 80.33 nM and 24.65 nM respectively in radioligand binding assays) and very low affinity for A3 Adenosine receptor (Ki =967.48 nM). It allows to perform cell visualization in fluorescence microscopy, confocal microscopy and high content system experiments. It is potentially suitable for other fluorescence-based assays.

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  • CELT-360

    Potent and partially selective hA1 Adenosine receptors fluorescent antagonist (646/662)

    Our potent and partially selective hA1 Adenosin receptor fluorescent antagonist shows affinity for hA1, hA2A and hA2B Adenosine receptors (Ki =8.60 nM, 98.38 nM, 72.24 and 231.01 nM respectively in radioligand binding assays). It allows to perform cell visualization in fluorescence microscopy, confocal microscopy and high content system experiments. It is potentially suitable for other fluorescence-based assays.

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  • CELT-300

    Potent and selective hA2A Adenosine receptor fluorescent ligand (646/662)

    Our hA2A Adenosine receptor fluorescent ligand shows high affinity and selectivity for hA2A receptor (Ki =8.35 nM for hA2A receptor in radioligand binding assay). It allows to perform cell visualization in fluorescence microscopy, confocal microscopy and high content system experiments. It is potentially suitable for other fluorescence-based assays.

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  • CELT-316

    Potent and selective hA2A Adenosine receptor fluorescent ligand (589/616)

    Our hA2A Adenosine receptor fluorescent ligand shows high affinity and selectivity for hA2A receptor (Ki =116.1 nM for hA2A receptor in radioligand binding assay). It allows to perform cell visualization in fluorescence microscopy, confocal microscopy and high content system experiments. It is potentially suitable for other fluorescence-based assays.

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  • CELT-327

    Potent hA2B/A3 Adenosine receptor fluorescent antagonist (589/616)

    Our hA2B/A3 Adenosine receptor fluorescent antagonist shows high affinity for hA2B and A3 receptor (Ki =35.6 nM and 45.7 nM respectively in radioligand binding assay). It allows to perform cell visualization in fluorescence microscopy, confocal microscopy and high content system experiments. It is potentially suitable for other fluorescence-based assays.

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  • CELT-171

    Potent and selective hA3 Adenosine receptor fluorescent antagonist (589/616)

    Our hA3 Adenosine receptor fluorescent antagonist shows a high affinity and selectivity for A3 receptor over the other receptor subtypes (Ki =6.13 nM for A3 receptor in radioligand binding assay). It allows to perform cell visualization in fluorescence microscopy, confocal microscopy and high content system experiments. It is potentially suitable for other fluorescence-based assays.

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  • CELT-402

    Potent h5HT2A Serotonin receptor fluorescent antagonist (589/616)

    Our h5HT2A Serotonin receptor fluorescent antagonist shows a high affinity for 5HT2A serotonin receptor (Ki =29.7 nM in radioligand binding assay).It allows to perform cell visualization in fluorescence microscopy, confocal microscopy and high content system experiments. It is potentially suitable for other fluorescence-based assays.

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  • CELT- 211

    Potent and selective h5HT2B Serotonin receptor fluorescent ligand (589/616)

    Our h5HT2B Serotonin receptor fluorescent ligand shows a high affinity for 5HT2B serotonin receptor and high selectivity over the other receptor subtypes (Ki =56.32 nM for 5HT2B receptor in radioligand binding assay).It allows to perform cell visualization in fluorescence microscopy, confocal microscopy and high content system experiments. It is potentially suitable for other fluorescence-based assays.

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  • CELT-335

    Potent CB1/CB2 Cannabinoids receptors fluorescent ligand (646/662)

    Our hCB cannabinoids receptors fluorescent ligand shows high affinity for hCB1/hCB2 cannabinoids receptor (Ki =44.8 nM and 7.4 nM , respectively in radioligand binding assay). It is suitable for HTRF binding assays as a valid alternative to radioligand binding assays. It allows to perform cell visualization in fluorescence microscopy, confocal microscopy and high content system experiments. It is potentially suitable for other fluorescence-based assays.

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  • CELT331

    Potent and selective hCB2 Cannabinoids receptors fluorescent ligand (646/662)

    Our hCB2 cannabinoids receptor fluorescent ligand shows high affinity for hCB2 cannabinoids receptor and selectivity over hCB1 (Ki =75.9 nM for hCB2 receptor in radioligand binding assay). It is suitable for HTRF binding assays as a valid alternative to radioligand binding assays. It allows to perform cell visualization in fluorescence microscopy, confocal and high content system experiments. It is potentially suitable for other fluorescence-based assays.

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  • CELT-195 (NIR)

    Potent M1 Muscarinic receptor fluorescent antagonist (748/776)

    Our M1 Muscarinic receptor fluorescent antagonist shows high affinity for M1 Muscrinic receptor (Ki =57.77 nM in radioligand binding assay). It allows to perform cell visualization in confocal microscopy and high content system experiments as a valid alternative to radioligand binding assays. It is potentially suitable for other fluorescence-based assays.

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