Adenosine Receptors
Celtarys is a market leader in developing fluorescent ligands for Adenosine Receptors, including A1, A2A, A2B, and A3 receptors. Our proprietary technology allows us to develop ligands with high specificity and affinity for these receptors, making them ideal for various applications, including receptor activation assays, tissue distribution studies, and more.
Our fluorescent ligands are designed to bind selectively to the Adenosine Receptor, allowing researchers to study the receptor’s signaling pathways and understand its role as a therapeutic target in the human body.
Our ligands are also highly effective in studying the nervous system, and their fluorescent properties allow for real-time imaging of receptor distribution and activation. They are versatile tools for studying G protein-coupled receptors and their interactions with ligands, including receptor antagonists.
At Celtarys, we are committed to providing you with the best products on the market for studying Adenosine Receptors, and we are constantly developing new solutions to meet your needs.
Showing all 10 results
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CELT- 480 hA3 Adenosine receptor fluorescent antagonist (646/662)
10ug vial that allows to prepare 70ml of 100nM working solution to test A3R.
432,00€
Working concentration might differ among assay designsView moreOur potent and selective hA3 Adenosine receptor fluorescent antagonist shows high affinity and selectivity for hA3 receptor (Ki =12 nM for hA3 receptor in radioligand binding assay). It allows to perform cell visualization in fluorescence microscopy, confocal microscopy and high content system experiments. It is potentially suitable for other fluorescence-based assays.
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CELT-298 Pan Adenosine receptors fluorescent antagonist (646/662)
10ug vial that allows to prepare 74ml of 100nM working solution to test A2AR.
432,00€
Working concentration might differ among assay designsView moreOur potent Pan Adenosine receptors fluorescent antagonist shows affinity for hA1, hA2A, hA2B and hA3 Adenosine receptors (Ki =20.9 nM, 171 nM, 44,7nM and 95.2 nM respectively in radioligand binding assays). It allows to perform cell visualization in fluorescence microscopy, confocal microscopy and high content system experiments. It is potentially suitable for other fluorescence-based assays.
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CELT-448 hA1 Adenosine receptor fluorescent antagonist (560/571)
10ug vial that allows to prepare 77ml of 100nM working solution to test A1R.
432,00€
Working concentration might differ among assay designsView morePotent and selective hA1 Adenosine receptors fluorescent antagonist (560/571)
Our potent and selective hA1 Adenosin receptor fluorescent antagonist shows affinity and selectivity for hA1, (Ki =26.2 nM in radioligand binding assays). It allows to perform cell visualization in fluorescence microscopy, confocal microscopy and high content system experiments. It is potentially suitable for other fluorescence-based assays.
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CELT-372 hA1/hA2b Adenosine receptors fluorescent antagonist (589/616)
10ug vial that allows to prepare 86ml of 100nM working solution to test A1R/A2R.
432,00€
Working concentration might differ among assay designsView moreOur potent hA1/A2B Adenosine receptor fluorescent antagonist shows affinity for hA1and hA2B Adenosine receptors (Ki =1.89 nMand 24.65 nM respectively in radioligand binding assays), intermediate affinity for A2A (Ki=80.33 nM) and very low affinity for A3 Adenosine receptor (Ki =967.48 nM). It allows to perform cell visualization in fluorescence microscopy, confocal microscopy and high content system experiments. It is potentially suitable for other fluorescence-based assays.
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CELT-360 hA1 Adenosine receptor fluorescent antagonist (646/662)
10ug vial that allows to prepare 78ml of 100nM working solution to test A1R.
432,00€
Working concentration might differ among assay designsView moreOur potent and partially selective hA1 Adenosine receptor fluorescent antagonist shows higher affinity for hA1 (Ki =8.60 nM) compared to hA2A, hA2B and hA3 Adenosine receptors (Ki= 98.38 nM, 72.24 and 231.01 nM respectively in radioligand binding assays). It allows to perform cell visualization in fluorescence microscopy, confocal microscopy and high content system experiments. It is potentially suitable for other fluorescence-based assays.
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CELT-300 hA2A Adenosine receptor fluorescent ligand (646/662)
10ug vial that allows to prepare 75ml of 100nM working solution to test A2AR
432,00€View moreOur potent and selective hA2A Adenosine receptor fluorescent ligand shows high affinity and selectivity for hA2A receptor (Ki =8.35 nM for hA2A receptor in radioligand binding assay). It allows to perform cell visualization in fluorescence microscopy, confocal microscopy and high content system experiments. It is potentially suitable for other fluorescence-based assays.
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CELT-316 hA2A Adenosine receptor fluorescent ligand (589/616)
10ug vial that allows to prepare 87ml of 100nM working solution to test A2AR.
432,00€
Working concentration might differ among assay designsView moreOur potent and selective hA2A Adenosine receptor fluorescent ligand shows high affinity and selectivity for hA2A receptor (Ki =116.1 nM for hA2A receptor in radioligand binding assay). It allows to perform cell visualization in fluorescence microscopy, confocal microscopy and high content system experiments. It is potentially suitable for other fluorescence-based assays.
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CELT-327 hA2B/A3 Adenosine receptor fluorescent antagonist (589/616)
10ug vial that allows to prepare 82ml of 100nM working solution to test A3R/A2BR.
432,00€
Working concentration might differ among assay designsView moreOur potent hA2B/A3 Adenosine receptor fluorescent antagonist shows high affinity for hA2B and A3 receptor (Ki =35.6 nM and 45.7 nM respectively in radioligand binding assay). It allows to perform cell visualization in fluorescence microscopy, confocal microscopy and high content system experiments. It is potentially suitable for other fluorescence-based assays.
More information and applications
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CELT-228 hA3 Adenosine receptor fluorescent antagonist (560/571)
10ug vial that allows to prepare 77ml of 100nM working solution to test A3R.
432,00€
Working concentration might differ among assay designsView moreOur potent and selective hA3 Adenosine receptor fluorescent antagonist shows high affinity for hA3 receptor and partial selectivity over the other receptor subtypes (Ki =52.7 nM for hA3 receptor in radioligand binding assay). It has been validated in Fluorescence Polarization binding assays as a valid alternative to radioligand binding assays.It allows to perform cell visualization in fluorescence microscopy, confocal microscopy and high content system experiments. It is potentially suitable for other fluorescence-based assays.
More information and applications
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CELT- 171 hA3 Adenosine receptor fluorescent antagonist (589/616)
10ug vial that allows to prepare 86ml of 100nM working solution to test A3R.
432,00€
Working concentration might differ among assay designsView moreOur potent and selective hA3 Adenosine receptor fluorescent antagonist shows a high affinity and selectivity for hA3 receptor over the other receptor subtypes (Ki =6.13 nM for A3 receptor in radioligand binding assay). It allows to perform cell visualization in fluorescence microscopy, confocal microscopy and high content system experiments. It is potentially suitable for other fluorescence-based assays.