Adenosine Receptors

Adenosine Receptors

Showing all 7 results

  • CELT-298

    Potent Pan Adenosine receptors fluorescent antagonist (646/662)

    Our Pan Adenosine receptors fluorescent antagonist shows affinity for hA1, hA2A, hA2B and hA3 Adenosine receptors (Ki =20.9 nM, 171 nM, 44,7nM and 95.2 nM respectively in radioligand binding assays). It allows to perform cell visualization in fluorescence microscopy, confocal microscopy and high content system experiments. It is potentially suitable for other fluorescence-based assays.

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  • CELT-372

    Potent and partially selective hA1 Adenosine receptors fluorescent antagonist (589/616)

    Our potent and partially selective hA1 Adenosin receptor fluorescent antagonist shows affinity for hA1, hA2A and hA2B Adenosine receptors (Ki =1.89 nM, 80.33 nM and 24.65 nM respectively in radioligand binding assays) and very low affinity for A3 Adenosine receptor (Ki =967.48 nM). It allows to perform cell visualization in fluorescence microscopy, confocal microscopy and high content system experiments. It is potentially suitable for other fluorescence-based assays.

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  • CELT-360

    Potent and partially selective hA1 Adenosine receptors fluorescent antagonist (646/662)

    Our potent and partially selective hA1 Adenosin receptor fluorescent antagonist shows affinity for hA1, hA2A and hA2B Adenosine receptors (Ki =8.60 nM, 98.38 nM, 72.24 and 231.01 nM respectively in radioligand binding assays). It allows to perform cell visualization in fluorescence microscopy, confocal microscopy and high content system experiments. It is potentially suitable for other fluorescence-based assays.

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  • CELT-300

    Potent and selective hA2A Adenosine receptor fluorescent ligand (646/662)

    Our hA2A Adenosine receptor fluorescent ligand shows high affinity and selectivity for hA2A receptor (Ki =8.35 nM for hA2A receptor in radioligand binding assay). It allows to perform cell visualization in fluorescence microscopy, confocal microscopy and high content system experiments. It is potentially suitable for other fluorescence-based assays.

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  • CELT-316

    Potent and selective hA2A Adenosine receptor fluorescent ligand (589/616)

    Our hA2A Adenosine receptor fluorescent ligand shows high affinity and selectivity for hA2A receptor (Ki =116.1 nM for hA2A receptor in radioligand binding assay). It allows to perform cell visualization in fluorescence microscopy, confocal microscopy and high content system experiments. It is potentially suitable for other fluorescence-based assays.

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  • CELT-327

    Potent hA2B/A3 Adenosine receptor fluorescent antagonist (589/616)

    Our hA2B/A3 Adenosine receptor fluorescent antagonist shows high affinity for hA2B and A3 receptor (Ki =35.6 nM and 45.7 nM respectively in radioligand binding assay). It allows to perform cell visualization in fluorescence microscopy, confocal microscopy and high content system experiments. It is potentially suitable for other fluorescence-based assays.

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  • CELT-171

    Potent and selective hA3 Adenosine receptor fluorescent antagonist (589/616)

    Our hA3 Adenosine receptor fluorescent antagonist shows a high affinity and selectivity for A3 receptor over the other receptor subtypes (Ki =6.13 nM for A3 receptor in radioligand binding assay). It allows to perform cell visualization in fluorescence microscopy, confocal microscopy and high content system experiments. It is potentially suitable for other fluorescence-based assays.

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