Cannabinoid Receptors

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  • CELT-335 hCB1/CB2 Cannabinoids receptors fluorescent ligand (646/662)

    10ug vial that allows to prepare 150ml of 100nM working solution to test CB1R/CB2R.

    Working concentration might differ among assay designs

    432,00

    Our potent hCB cannabinoids receptors fluorescent ligand shows high affinity for hCB1/CB2 cannabinoids receptor (Ki =44.8 nM and 7.4 nM , respectively in radioligand binding assay). It has been validated in High Content Screening assays and it is suitable also for HTRF binding assays as a valid alternative to radioligand binding assays. It allows to perform cell visualization in fluorescence microscopy and it is potentially suitable for other fluorescence-based assays.

    More information and applications

    https://www.sciencedirect.com/science/article/pii/S1043661821005545?via%3Dihub

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  • CELT-331 hCB2 Cannabinoids receptor fluorescent ligand (646/662)

    Our potent and selective hCB2 cannabinoids receptor fluorescent ligand shows high affinity for hCB2 cannabinoids receptor and selectivity over hCB1 (Ki =75.9 nM for hCB2 receptor in radioligand binding assay). It is suitable for HTRF binding assays as a valid alternative to radioligand binding assays. It allows to perform cell visualization in fluorescence microscopy, confocal and high content system experiments. It is potentially suitable for other fluorescence-based assays.

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