Dopamine D2 Receptor Family
At Celtarys, we offer a comprehensive range of fluorescent ligands for dopamine receptors, including D2 and D3 receptors. Our proprietary technology enables us to develop ligands with high affinity and specificity, making them ideal for a variety of applications, including binding assays, fluorescence-based assays, and more.
Showing all 7 results
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CELT- 174 hD2 Dopamine receptor fluorescent antagonist (589/616)
Our potent hD2 dopamine receptor fluorescent antagonist is available in a 10ug vial, allowing you to prepare 73ml of 100nM working solution to test D2R.
432,00€
Our CELT-174 product has been specifically designed to meet the needs of researchers in a variety of fields, enabling the study of D2 dopamine receptors with greater accuracy and precisionView moreOur potent and selective hD2 Dopamine receptor fluorescent antagonist shows high affinity for hD2 receptor and selectivity over the other receptor subtypes (Ki =1.06 nM for hD2 receptor in radioligand binding assay). It allows to perform cell visualization in fluorescence microscopy, confocal microscopy and high content system experiments. It is potentially suitable for other fluorescence-based assays.
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CELT- 426 hD2 Dopamine receptor fluorescent antagonist (560/571)
Our CELT-426 product is available in a 10ug vial that allows you to prepare 67ml of 100nM working solution to test D2R.
432,00€
It has been specifically designed for high potency and selectivity, demonstrating a high affinity for D2 receptors and may be suitable for fluorescence-based assaysView moreOur potent and partially selective hD2 Dopamine receptor fluorescent antagonist shows high affinity for hD2 receptor and partial selectivity over the other receptor subtypes (Ki =89.3 nM for hD2 receptor in radioligand binding assay). It has been validated in Fluorescence Polarization binding assays as a valid alternative to radioligand binding assays.It allows to perform cell visualization in fluorescence microscopy, confocal microscopy and high content system experiments. It is potentially suitable for other fluorescence-based assays.
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CELT- 419 hD3 Dopamine receptor fluorescent ligand (560/571)
Our CELT-419 product is available in a 10ug vial that allows you to prepare 74ml of 100nM working solution to test D3R.
432,00€
It has been specifically designed to target the D3 dopamine receptor, making it an ideal tool for researchers performing cell visualization in fluorescence microscopyView moreOur potent and partially selective hD3 Dopamine receptor fluorescent ligand shows high affinity for hD3 receptor and partial selectivity over the other receptor subtypes (Ki =65.6 nM for hD3 receptor in radioligand binding assay). It has been validated in Fluorescence Polarization binding assays as a valid alternative to radioligand binding assays.It allows to perform cell visualization in fluorescence microscopy, confocal microscopy and high content system experiments. It is potentially suitable for other fluorescence-based assays.
More information and applications
https://www.frontiersin.org/articles/10.3389/fmolb.2023.1119157/full
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CELT-240 hD2/D3 Dopamine receptors fluorescent ligand (589/616)
Our CELT-240 product is available in a 10ug vial that allows you to prepare 78ml of 100nM working solution to test D2R/D3R.
432,00€
It demonstrates high potency and selectivity, making it a valuable tool for researchers interested in studying the D2 and D3 receptorsView moreOur potent hD3/D2 Dopamine receptors fluorescent ligand shows high affinity for hD2 and hD3 receptors (Ki =2.34 nM and 2.14 nM respectively in radioligand binding assays) and selectivity over D4 dopamine receptor. It allows to perform cell visualization in fluorescence microscopy, confocal microscopy and high content system experiments. It is potentially suitable for other fluorescence-based assays.
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CELT-241 hD2/D3 Dopamine receptors fluorescent ligand (646/662)
Our CELT-241 product is available in a 10ug vial that allows you to prepare 68ml of 100nM working solution to test D2R/D3R.
432,00€
It demonstrates high potency and selectivity, making it a valuable tool for researchers interested in studying D2 and D3 receptorsView moreOur potent hD2/D3 Dopamine receptors fluorescent ligand shows a high affinity for hD2 and hD3 receptors (Ki = 5.22 nM and 4.77 nM respectively in radioligand binding assays) nd selectivity over D4 dopamine receptor. It allows to perform cell visualization in fluorescence microscopy, confocal microscopy and high content system experiments. It is potentially suitable for other fluorescence-based assays.
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CELT-429 hD3 Dopamine receptor fluorescent ligand (589/616)
Our CELT-429 product is available in a 10ug vial that allows you to prepare 78ml of 100nM working solution to test D3R.
432,00€
It demonstrates high potency and selectivity, making it a valuable tool for researchers interested in studying the role of D3 receptors in various physiological and pathological conditionsView moreOur potent and selective hD3 Dopamine receptors fluorescent ligand shows a high affinity for hD3 receptors (Ki = 75.4 nM in radioligand binding assays) and selectivity over D3 and D4 dopamine receptor. It allows to perform cell visualization in fluorescence microscopy, confocal microscopy and high content system experiments. It is potentially suitable for other fluorescence-based assays.
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CELT-175 hD2 Dopamine receptor fluorescent antagonist (748/776)
Our CELT-175 product is available in a 10ug vial that allows you to prepare 63ml of 100nM working solution to test D2R.
432,00€
It has been specifically designed for high potency and selectivity, demonstrating a high affinity for D2 receptors and may be suitable for fluorescence-based assaysView moreOur potent and selective hD2 Dopamine receptor fluorescent antagonist shows high affinity for hD2 receptor and selectivity over the other receptor subtypes (Ki =3.15 nM for hD2 receptor and Ki =294.6 nM and Ki =220.3 nM for D3 and D4 receptor, respectively, in radioligand binding assay). It allows to perform cell visualization in fluorescence microscopy, confocal microscopy and high content system experiments. It is potentially suitable for other fluorescence-based assays.