CELT- 402 h5HT2A/5HT2C Serotonin receptor fluorescent antagonist (589/616)
7 January 2021
CELT- 419 hD3 Dopamine receptor fluorescent ligand (560/571)
15 July 2021

CELT- 426 hD2 Dopamine receptor fluorescent antagonist (560/571)

10ug vial that allows to prepare 37ml of 100nM working solution to test D2R.

Working concentration might differ among assay designs


Our potent and partially selective hD2 Dopamine receptor fluorescent antagonist shows high affinity for hD2 receptor and partial selectivity over the other receptor subtypes (Ki =89.3 nM for hD2 receptor in radioligand binding assay). It has been validated in Fluorescence Polarization binding assays as a valid alternative to radioligand binding assays.It allows to perform cell visualization in fluorescence microscopy, confocal microscopy and high content system experiments. It is potentially suitable for other fluorescence-based assays.