Adrenergic Receptors

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  • CELT-130 hα1 adrenergic receptor fluorescent antagonist (646/662)

    10ug vial that allows to prepare 150ml of 100nM working solution to test alpha1AR.

    Working concentration might differ among assay designs

    432,00

    Our potent and selective hα1A  adrenergic receptor fluorescent antagonist shows high affinity for α1A adrenergic receptor (Ki =28.3 nM measured in radioligand binding assay) and selectivity over  α2A (Ki =1081 nM measured in radioligand binding assay). It is potentially suitable for fluorescence-based assays such as confocal microscopy or high content screening.

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  • CELT-133 hα1 adrenergic receptor fluorescent antagonist (560/571)

    10ug vial that allows to prepare 830ml of 100nM working solution to test alpha1AR.

    Working concentration might differ among assay designs

    432,00

    Our potent and selective hα1A  adrenergic receptor fluorescent antagonist shows high affinity for alpha 1 adrenergic receptor (Ki =5 nM measured in radioligand binding assay) and selectivity over  α2A (15% of displacement at 1 μM in radioligand binding assay). It is potentially suitable for fluorescence-based assays such as confocal microscopy, high content screening or fluorescence polarization.

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