Adrenergic Receptors

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  • CELT-130 hα1 adrenergic receptor fluorescent antagonist (646/662)

    Our potent and selective hα1A  adrenergic receptor fluorescent antagonist shows high affinity for α1A adrenergic receptor (Ki =28.3 nM measured in radioligand binding assay) and selectivity over  α2A (Ki =1081 nM measured in radioligand binding assay). It is potentially suitable for fluorescence-based assays such as confocal microscopy or high content screening.

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  • CELT-133 hα1 adrenergic receptor fluorescent antagonist (560/571)

    Our potent and selective hα1A  adrenergic receptor fluorescent antagonist shows high affinity for alpha 1 adrenergic receptor (Ki =5 nM measured in radioligand binding assay) and selectivity over  α2A (15% of displacement at 1 μM in radioligand binding assay). It is potentially suitable for fluorescence-based assays such as confocal microscopy, high content screening or fluorescence polarization.

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