Adrenergic Receptors

At Celtarys, we offer a comprehensive range of fluorescent ligands α1a adrenergic receptors. Our proprietary technology enables us to develop ligands with high affinity and specificity, making them ideal for a variety of applications, including receptor activation assays and more.

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  • CELT-130 hα1 adrenergic receptor fluorescent antagonist (646/662)

    10ug vial that allows to prepare 83ml of 100nM working solution to test alpha1AR.

    Working concentration might differ among assay designs
    Our CELT-130 product has been developed to meet the needs of researchers in a variety of fields, enabling the study of alpha1a adrenergic receptors with greater accuracy and precision.

    432,00

    Our potent and selective hα1A  adrenergic receptor fluorescent antagonist shows high affinity for α1A adrenergic receptor (Ki =28.3 nM measured in radioligand binding assay) and selectivity over  α2A (Ki =1081 nM measured in radioligand binding assay). It is potentially suitable for fluorescence-based assays such as confocal microscopy or high content screening.

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  • CELT-133 hα1 adrenergic receptor fluorescent antagonist (560/571)

    This product is available in a 10ug vial that allows you to prepare 83ml of 100nM working solution to test alpha1AR.

    The working concentration might differ among assay designs
    Our CELT-133 ligand has been specifically designed for high potency and selectivity. It has a high affinity for α1 receptors and may be suitable for fluorescence-based assays.

    432,00

    Our potent and selective hα1A  adrenergic receptor fluorescent antagonist shows high affinity for alpha 1 adrenergic receptor (Ki =5 nM measured in radioligand binding assay) and selectivity over  α2A (15% of displacement at 1 μM in radioligand binding assay). It is potentially suitable for fluorescence-based assays such as confocal microscopy, high content screening or fluorescence polarization.

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