Muscarinic Receptors

At Celtarys, we offer a comprehensive range of fluorescent ligands for muscarinic receptors, including M1 and M2 receptors. Our proprietary technology enables us to develop ligands with high affinity and specificity, making them ideal for a variety of applications, including binding assays.

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  • CELT-249 hM1/M2 Muscarinic Receptor fluorescent antagonist (589/616)

    10ug vial that allows to prepare 82ml of 100nM working solution to test M1/M2 Muscarinic Receptor.

    Working concentration might differ among assay designs

    432,00

    Our CELT-249 ligand is a highly potent fluorescent antagonist developed for hM1R and hM2R testing with a Ki of 133 nM and 11.5 nM, respectively in radioligand binding assay. The product comes in a 10ug vial that enables the preparation of 82ml of 100nM working solution to test M1R/M2R. Our fluorescent antagonist is ideal for visualization in confocal microscopy and high-content system experiments. Our CELT-249 ligand is potentially suitable for other fluorescence-based assays

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  • CELT-195 hM1/M2 Muscarinic receptor fluorescent antagonist (748/776)

    10ug vial that allows to prepare 73ml of 100nM working solution to test M1R/M2R.

    Working concentration might differ among assay designs

    432,00

    Our CELT-195 ligand is a highly potent fluorescent antagonist developed for M1R and M2R testing with a Ki of 57.77 nM and 37.7 nM, respectively in radioligand binding assay. The product comes in a 10ug vial that enables the preparation of 95ml of 100nM working solution to test M1R/M2R. Our fluorescent antagonist is ideal for visualization in confocal microscopy and high-content system experiments. Our CELT-195 ligand is potentially suitable for other fluorescence-based assays.

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