Products
CELT-300 hA2A Adenosine receptor fluorescent ligand (646/662)
24 December 2020CELT-372 hA1/hA2b Adenosine receptors fluorescent antagonist (589/616)
24 December 2020
CELT-360 hA1 Adenosine receptor fluorescent antagonist (646/662)
10ug vial that allows to prepare 78ml of 100nM working solution to test A1R.
Working concentration might differ among assay designs
432,00€
Our potent and partially selective hA1 Adenosine receptor fluorescent antagonist shows higher affinity for hA1 (Ki =8.60 nM) compared to hA2A, hA2B and hA3 Adenosine receptors (Ki= 98.38 nM, 72.24 and 231.01 nM respectively in radioligand binding assays). It allows to perform cell visualization in fluorescence microscopy, confocal microscopy and high content system experiments. It is potentially suitable for other fluorescence-based assays.
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CELT-298 Pan Adenosine receptors fluorescent antagonist (646/662)
10ug vial that allows to prepare 74ml of 100nM working solution to test A2AR.
432,00€
Working concentration might differ among assay designsView moreOur potent Pan Adenosine receptors fluorescent antagonist shows affinity for hA1, hA2A, hA2B and hA3 Adenosine receptors (Ki =20.9 nM, 171 nM, 44,7nM and 95.2 nM respectively in radioligand binding assays). It allows to perform cell visualization in fluorescence microscopy, confocal microscopy and high content system experiments. It is potentially suitable for other fluorescence-based assays.
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CELT-448 hA1 Adenosine receptor fluorescent antagonist (560/571)
10ug vial that allows to prepare 77ml of 100nM working solution to test A1R.
432,00€
Working concentration might differ among assay designsView morePotent and selective hA1 Adenosine receptors fluorescent antagonist (560/571)
Our potent and selective hA1 Adenosin receptor fluorescent antagonist shows affinity and selectivity for hA1, (Ki =26.2 nM in radioligand binding assays). It allows to perform cell visualization in fluorescence microscopy, confocal microscopy and high content system experiments. It is potentially suitable for other fluorescence-based assays.
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CELT-228 hA3 Adenosine receptor fluorescent antagonist (560/571)
10ug vial that allows to prepare 77ml of 100nM working solution to test A3R.
432,00€
Working concentration might differ among assay designsView moreOur potent and selective hA3 Adenosine receptor fluorescent antagonist shows high affinity for hA3 receptor and partial selectivity over the other receptor subtypes (Ki =52.7 nM for hA3 receptor in radioligand binding assay). It has been validated in Fluorescence Polarization binding assays as a valid alternative to radioligand binding assays.It allows to perform cell visualization in fluorescence microscopy, confocal microscopy and high content system experiments. It is potentially suitable for other fluorescence-based assays.
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