CELT-195 hM1/M2 Muscarinic receptor fluorescent antagonist (748/776)
24 December 2020

CELT- 171 hA3 Adenosine receptor fluorescent antagonist (589/616)

10ug vial that allows to prepare 86ml of 100nM working solution to test A3R.

Working concentration might differ among assay designs


Our potent and selective hA3 Adenosine receptor fluorescent antagonist shows a high affinity and selectivity for hA3 receptor over the other receptor subtypes (Ki =6.13 nM for A3 receptor in radioligand binding assay). It allows to perform cell visualization in fluorescence microscopy, confocal microscopy and high content system experiments. It is potentially suitable for other fluorescence-based assays.