Products
CELT-448 hA1 Adenosine receptor fluorescent antagonist (560/571)
15 July 2021LUXendin551 GLP1 receptor (GLP1R) fluorescent antagonist (551/576) (CELT-111)
27 September 2021
CELT-228 hA3 Adenosine receptor fluorescent antagonist (560/571)
10ug vial that allows to prepare 77ml of 100nM working solution to test A3R.
Working concentration might differ among assay designs
432,00€
Our potent and selective hA3 Adenosine receptor fluorescent antagonist shows high affinity for hA3 receptor and partial selectivity over the other receptor subtypes (Ki =52.7 nM for hA3 receptor in radioligand binding assay). It has been validated in Fluorescence Polarization binding assays as a valid alternative to radioligand binding assays.It allows to perform cell visualization in fluorescence microscopy, confocal microscopy and high content system experiments. It is potentially suitable for other fluorescence-based assays.
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CELT-300 hA2A Adenosine receptor fluorescent ligand (646/662)
10ug vial that allows to prepare 75ml of 100nM working solution to test A2AR
432,00€View moreOur potent and selective hA2A Adenosine receptor fluorescent ligand shows high affinity and selectivity for hA2A receptor (Ki =8.35 nM for hA2A receptor in radioligand binding assay). It allows to perform cell visualization in fluorescence microscopy, confocal microscopy and high content system experiments. It is potentially suitable for other fluorescence-based assays.
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CELT-360 hA1 Adenosine receptor fluorescent antagonist (646/662)
10ug vial that allows to prepare 78ml of 100nM working solution to test A1R.
432,00€
Working concentration might differ among assay designsView moreOur potent and partially selective hA1 Adenosine receptor fluorescent antagonist shows higher affinity for hA1 (Ki =8.60 nM) compared to hA2A, hA2B and hA3 Adenosine receptors (Ki= 98.38 nM, 72.24 and 231.01 nM respectively in radioligand binding assays). It allows to perform cell visualization in fluorescence microscopy, confocal microscopy and high content system experiments. It is potentially suitable for other fluorescence-based assays.
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CELT-327 hA2B/A3 Adenosine receptor fluorescent antagonist (589/616)
10ug vial that allows to prepare 82ml of 100nM working solution to test A3R/A2BR.
432,00€
Working concentration might differ among assay designsView moreOur potent hA2B/A3 Adenosine receptor fluorescent antagonist shows high affinity for hA2B and A3 receptor (Ki =35.6 nM and 45.7 nM respectively in radioligand binding assay). It allows to perform cell visualization in fluorescence microscopy, confocal microscopy and high content system experiments. It is potentially suitable for other fluorescence-based assays.
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