CELT- 171 hA3 Adenosine receptor fluorescent antagonist (589/616)
21 June 2020
CELT-331 hCB2 Cannabinoids receptor fluorescent ligand (646/662)
24 December 2020

CELT-195 hM1/M2 Muscarinic receptor fluorescent antagonist (748/776)

10ug vial that allows to prepare 73ml of 100nM working solution to test M1R/M2R.

Working concentration might differ among assay designs


Our CELT-195 ligand is a highly potent fluorescent antagonist developed for M1R and M2R testing with a Ki of 57.77 nM and 37.7 nM, respectively in radioligand binding assay. The product comes in a 10ug vial that enables the preparation of 95ml of 100nM working solution to test M1R/M2R. Our fluorescent antagonist is ideal for visualization in confocal microscopy and high-content system experiments. Our CELT-195 ligand is potentially suitable for other fluorescence-based assays.