CELT- 171 hA3 Adenosine receptor fluorescent antagonist (589/616)
21 June 2020
CELT-331 hCB2 Cannabinoids receptor fluorescent ligand (646/662)
24 December 2020

CELT-195 hM1/M2 Muscarinic receptor fluorescent antagonist (748/776)

10ug vial that allows to prepare 95ml of 100nM working solution to test M1R/M2R.

Working concentration might differ among assay designs


Our potent hM1/hM2 Muscarinic receptor fluorescent antagonist shows high affinity for hM1 and hM2 Muscarinic receptors (Ki =57.77 nM and 37,7 nM respectively in radioligand binding assay). It allows to perform cell visualization in confocal microscopy and high content system experiments as a valid alternative to radioligand binding assays. It is potentially suitable for other fluorescence-based assays.