CELT-195 hM1/M2 Muscarinic receptor fluorescent antagonist (748/776)
24 December 2020
CELT-335 hCB1/CB2 Cannabinoids receptors fluorescent ligand (646/662)
24 December 2020

CELT-331 hCB2 Cannabinoids receptor fluorescent ligand (646/662)

Our potent and selective hCB2 cannabinoids receptor fluorescent ligand shows high affinity for hCB2 cannabinoids receptor and selectivity over hCB1 (Ki =75.9 nM for hCB2 receptor in radioligand binding assay). It is suitable for HTRF binding assays as a valid alternative to radioligand binding assays. It allows to perform cell visualization in fluorescence microscopy, confocal and high content system experiments. It is potentially suitable for other fluorescence-based assays.