Products

CELT-130 hα1 adrenergic receptor fluorescent antagonist (646/662)
4 October 2022

CELT-133 hα1 adrenergic receptor fluorescent antagonist (560/571)

Our potent and selective hα1A  adrenergic receptor fluorescent antagonist shows high affinity for alpha 1 adrenergic receptor (Ki =5 nM measured in radioligand binding assay) and selectivity over  α2A (15% of displacement at 1 μM in radioligand binding assay). It is potentially suitable for fluorescence-based assays such as confocal microscopy, high content screening or fluorescence polarization.