Binding Assays

25 May 2026
Fluorescence Polarization Binding Assays for E3 Ligases in Targeted Protein Degradation (TPD) Programs

Fluorescence Polarization Binding Assays for E3 Ligases in Targeted Protein Degradation (TPD) Programs

Targeted protein degradation (TPD) has reshaped drug discovery by eliminating disease-driving proteins through the cell’s own degradation systems, rather than merely blocking their activity. PROTACs (bifunctional […]