Identifying new E3 Ubiquitin ligase ligands for new PROTACs design is a key element that can improve selective proteasomal-dependent degradation of proteins of interest involved in many pathological processes such as cancer, chronic anaemia, and ischemia.
Our fluorescent probes for VHL and CRBN E3 ligase are powerful tools both for compound screening for new E3ligase ligands and for PROTACs analysis, suitable for in vitro microscopy, binding assays such as TR-FRET competition assays.
-
CELT-077 CRBN E3 ligase fluorescent ligand (589/616)
For research use only10 µg vial that allows to prepare 46.2 mL of 200 nM working solution.
476,00€
Working concentration might differ among assay designsView moreProduct on backorder. Contact us at info@celtarys.com for an estimated delivery date.
-
CELT-081 CRBN E3 ligase fluorescent ligand (646/662)
For research use only10 µg vial that allows to prepare 39.4 mL of 200 nM working solution.
476,00€
Working concentration might differ among assay designsView moreProduct on backorder. Contact us at info@celtarys.com for an estimated delivery date.
-
CELT-504 VHL E3 ligase fluorescent ligand (564/570)
For research use only10 µg vial that allows to prepare 47 mL of 200 nM working solution.
476,00€ View more
Working concentration might differ among assay designs -
CELT-050 VHL E3 ligase fluorescent ligand (646/662)
For research use only10 µg vial that allows to prepare 33.2 mL of 200 nM working solution.
476,00€
Working concentration might differ among assay designsView moreProduct on backorder. Contact us at info@celtarys.com for an estimated delivery date.
Do you want more information?
We are ready to support your challenges