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CELT-360 hA1 adenosine receptor fluorescent antagonist (646/662) For research use only

CHO cells expressing the human A1 receptor labelled with (A) 40 nM CELT-360, (B) 20 nM CELT-360 and (C) 10 nM CELT-360. Competition binding assay with CHO cells expressing the human A1 receptor labelled with (D) 40 nM CELT-360 and Hoechst 33342, (E) 40 nM CELT-360 and Hoechst 33342 preincubated with 10 µM XAC and (F) Hoechst 33342.

Our potent and partially selective hA₁ adenosine receptor fluorescent antagonist shows higher affinity for hA₁ (K_i = 8.60 nM) compared to hA_2A, hA_2B and hA₃ adenosine receptors (K_i = 98.38 nM, 72.24 nM and 231.01 nM respectively in radioligand binding assays). It allows to perform cell visualization in fluorescence microscopy, confocal microscopy and high content system experiments. It is potentially suitable for other fluorescence-based assays.

CELT-360 hA1 adenosine receptor fluorescent antagonist (646/662)
_{For research use only}

Name: CELT-360 hA1 adenosine receptor fluorescent antagonist (646/662) For research use only - Celtarys
Price: 476.00 EUR
Availability: InStock

10 µg vial can be used to prepare 78.89 µL of a 100 µM stock solution, providing enough volume for 7 assays at a working concentration of 100 nM.
Please note that the required concentration may vary depending on the specific assay design.

476,00€

In stock

Category: Adenosine Receptors

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More information and contact in info@celtarys.com

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CELT-360 hA1 adenosine receptor fluorescent antagonist (646/662) For research use only

10 µg vial can be used to prepare 78.89 µL of a 100 µM stock solution, providing enough volume for 7 assays at a working concentration of 100 nM.Please note that the required concentration may vary depending on the specific assay design.

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10 µg vial can be used to prepare 78.89 µL of a 100 µM stock solution, providing enough volume for 7 assays at a working concentration of 100 nM.
Please note that the required concentration may vary depending on the specific assay design.

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Please note that the required concentration may vary depending on the specific assay design.

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10 µg vial can be used to prepare 87.10 µL of a 100 µM stock solution, providing enough volume for 8 assays at a working concentration of 100 nM.
Please note that the required concentration may vary depending on the specific assay design.

CELT-372 hA1/hA2B adenosine receptors fluorescent antagonist (589/616)
_{For research use only}

10 µg vial can be used to prepare 85.68 µL of a 100 µM stock solution, providing enough volume for 8 assays at a working concentration of 100 nM.
Please note that the required concentration may vary depending on the specific assay design.