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CELT-228 hA3 adenosine receptor fluorescent antagonist (560/571) For research use only

Specific A3AR labelling in a panel of cell lines. Representative images of HeLa-A3, HCT116, SW480 and SW620 cells labelled with 250 nM CELT-228, and counterstained with CellTracker Green.

Our potent and selective hA₃ adenosine receptor fluorescent antagonist shows high affinity for hA₃ receptor and partial selectivity over the other receptor subtypes (K_i = 52.7 nM for hA₃ receptor in radioligand binding assay). It has been validated in Fluorescence Polarization binding assays as a valid alternative to radioligand binding assays. It allows to perform cell visualization in fluorescence microscopy, confocal microscopy and high content system experiments. It is potentially suitable for other fluorescence-based assays.

More information and applications

Article: Identification of A2BAR as a potential target in colorectal cancer using novel fluorescent GPCR ligands

Article: Exploring Non-orthosteric Interactions with a Series of Potent and Selective A3 Antagonists

CELT-228 hA3 adenosine receptor fluorescent antagonist (560/571)
_{For research use only}

Name: CELT-228 hA3 adenosine receptor fluorescent antagonist (560/571) For research use only - Celtarys
Price: 476.00 EUR
Availability: InStock

10 µg vial can be used to prepare 77.25 µL of a 100 µM stock solution, providing enough volume for 7 assays at a working concentration of 100 nM.
Please note that the required concentration may vary depending on the specific assay design.

476,00€

Product on backorder. Contact us at info@celtarys.com for an estimated delivery date.

Available on back-order

Category: Adenosine Receptors

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More information and applications

CELT-228 hA3 adenosine receptor fluorescent antagonist (560/571) For research use only

10 µg vial can be used to prepare 77.25 µL of a 100 µM stock solution, providing enough volume for 7 assays at a working concentration of 100 nM.Please note that the required concentration may vary depending on the specific assay design.

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CELT-228 hA3 adenosine receptor fluorescent antagonist (560/571)
_{For research use only}

10 µg vial can be used to prepare 77.25 µL of a 100 µM stock solution, providing enough volume for 7 assays at a working concentration of 100 nM.
Please note that the required concentration may vary depending on the specific assay design.

CELT-372 hA1/hA2B adenosine receptors fluorescent antagonist (589/616)
_{For research use only}

10 µg vial can be used to prepare 85.68 µL of a 100 µM stock solution, providing enough volume for 8 assays at a working concentration of 100 nM.
Please note that the required concentration may vary depending on the specific assay design.

CELT-298 PAN adenosine receptors fluorescent antagonist (646/662)
_{For research use only}

10 µg vial can be used to prepare 74.10 µL of a 100 µM stock solution, providing enough volume for 7 assays at a working concentration of 100 nM.
Please note that the required concentration may vary depending on the specific assay design.

CELT-464 hA2A adenosine receptor fluorescent antagonist (575/590)
_{For research use only}

10 µg vial can be used to prepare 89.85 µL of a 100 µM stock solution, providing enough volume for 8 assays at a working concentration of 100 nM.
Please note that the required concentration may vary depending on the specific assay design.

CELT-300 hA2A adenosine receptor fluorescent ligand (646/662)
_{For research use only}

10 µg vial can be used to prepare 75.72 µL of a 100 µM stock solution, providing enough volume for 7 assays at a working concentration of 100 nM.
Please note that the required concentration may vary depending on the specific assay design.