Our potent and selective hα1A  adrenergic receptor fluorescent antagonist shows high affinity for α1A adrenergic receptor (Ki =28.3 nM measured in radioligand binding assay) and selectivity over  α2A (Ki =1081 nM measured in radioligand binding assay). It is potentially suitable for fluorescence-based assays such as confocal microscopy or high content screening.

CELT-130 hα1 adrenergic receptor fluorescent antagonist (646/662)

10ug vial that allows to prepare 83ml of 100nM working solution to test alpha1AR.

Working concentration might differ among assay designs
Our CELT-130 product has been developed to meet the needs of researchers in a variety of fields, enabling the study of alpha1a adrenergic receptors with greater accuracy and precision.

432,00