Products

CELT-175 hD2 Dopamine receptor fluorescent antagonist (748/776)
14 March 2022
CELT-133 hα1 adrenergic receptor fluorescent antagonist (560/571)
4 October 2022

CELT-130 hα1 adrenergic receptor fluorescent antagonist (646/662)

10ug vial that allows to prepare 150ml of 100nM working solution to test alpha1AR.

Working concentration might differ among assay designs

432,00

Our potent and selective hα1A  adrenergic receptor fluorescent antagonist shows high affinity for α1A adrenergic receptor (Ki =28.3 nM measured in radioligand binding assay) and selectivity over  α2A (Ki =1081 nM measured in radioligand binding assay). It is potentially suitable for fluorescence-based assays such as confocal microscopy or high content screening.