Products

CELT-175 hD2 Dopamine receptor fluorescent antagonist (748/776)
14 March 2022
CELT-133 hα1 adrenergic receptor fluorescent antagonist (560/571)
4 October 2022

CELT-130 hα1 adrenergic receptor fluorescent antagonist (646/662)

Our potent and selective hα1A  adrenergic receptor fluorescent antagonist shows high affinity for α1A adrenergic receptor (Ki =28.3 nM measured in radioligand binding assay) and selectivity over  α2A (Ki =1081 nM measured in radioligand binding assay). It is potentially suitable for fluorescence-based assays such as confocal microscopy or high content screening.