Products
CELT-175 hD2 Dopamine receptor fluorescent antagonist (748/776)
14 March 2022CELT-133 hα1 adrenergic receptor fluorescent antagonist (560/571)
4 October 2022
CELT-130 hα1 adrenergic receptor fluorescent antagonist (646/662)
10ug vial that allows to prepare 150ml of 100nM working solution to test alpha1AR.
Working concentration might differ among assay designs
432,00€
Our potent and selective hα1A adrenergic receptor fluorescent antagonist shows high affinity for α1A adrenergic receptor (Ki =28.3 nM measured in radioligand binding assay) and selectivity over α2A (Ki =1081 nM measured in radioligand binding assay). It is potentially suitable for fluorescence-based assays such as confocal microscopy or high content screening.
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CELT-133 hα1 adrenergic receptor fluorescent antagonist (560/571)
10ug vial that allows to prepare 830ml of 100nM working solution to test alpha1AR.
432,00€
Working concentration might differ among assay designsView moreOur potent and selective hα1A adrenergic receptor fluorescent antagonist shows high affinity for alpha 1 adrenergic receptor (Ki =5 nM measured in radioligand binding assay) and selectivity over α2A (15% of displacement at 1 μM in radioligand binding assay). It is potentially suitable for fluorescence-based assays such as confocal microscopy, high content screening or fluorescence polarization.